Clomiphene citrate – this is a non-steroidal drug synthetic origin, its characteristics is classified as an antiestrogen. This drug has received the widest dissemination in medicine, and in heavy sports. For example, in medical practice used in quality Clomiphene ovulation stimulator.
With partial structural similarity with the hormone estrogen, antiestrogen clomiphene citrate can bind to estrogen receptors in the hypothalamus. Due to this there is a large production of gonadotropins FSH and LH, which in turn activates the secretion of the hormone testosterone in men and estrogen in women.
Clomiphene citrate in sports and medicine
This anti-estrogen is very specific and can have positive effects on multiple systems of the human body. For example, clomiphene citrate and analogs thereof (Clomid, etc.) can help women cope with ovarian dysfunction or normalize their work with minor deviations. The fact that many women are not able to get pregnant, there is disruption of ovulation. Among women with ovulation disorders distinguish patients with ovarian syndrome poltkistoznyh, and patients with amenorrhea. The drug is clomiphene citrate, after identifying the causes ovulation disorders can help overcome both the first and second disease, but only in the preparation of calibrated therapeutic course.
Clomid bodybuilding drug became renowned as clomiphene and similar preparations from other manufacturers. But as the drug gradually replacing their competitors. Although tablets efficiency remains constantly high.
Clomiphene Citrate Tablets are considered to be a potent drug and is rarely used for a long time. It is also important that their effectiveness depends on the time of receipt. In most cases, to determine the ovulation takes a blood sample and measure the temperature. The drug is Clomiphene Citrate starts to be used only after passing all the tests: prepared course of medication with the exact dosage, use of time, frequency and duration. Typically reception starts on the fifth day of the cycle and lasts for 3-6 cycles.
Has the anti-estrogen and contraindications for use. Thus, the drug clomiphene citrate can not be used during pregnancy or in the presence of ovarian cysts (before treatment the woman is obliged to pass the “ultrasound” in order to avoid an increase in the ovaries). Also, the anti-estrogen should not be used during vaginal bleeding or disorders of the liver.
It is worth noting that despite widespread in medical practice, for men Clomiphene Citrate is not the most reliable means, when it comes to the treatment of infertility. The reason for this is the small study of the impact of the drug on the male body. Yes, it is known that taking Clomid and similar means increases the secretion of LH and FSH, which has a positive effect on testosterone levels. However, the drug affects the genitals – unknown to the end. All studies on this subject were conducted on individual patients and only for a few months. Therefore, a reliable source of information, they can not be.
And that’s where Clomiphene Citrate is regularly used by men and at the same time efficiently, it is in bodybuilding. By the reception of the pharmacological agent is equally often used, as professional athletes and young athletes. The main advantage of the preparation in heavy sports is that it, in contrast to steroid hormones and does not reduce the natural testosterone concentration. On the contrary, Clomiphene citrate as used in the sport (in the appropriate “sports” doses), leads to a surge of LH, which increases levels of the male sex hormone.
Also Clomiphene Citrate can be used to neutralize the male gynecomastia that arises as a result of taking steroids. It is proved that all drugs have anabolic androgenic properties, albeit to varying degrees. In some cases, steroids promote the formation of estrogen in the male body (via the aromatase enzyme is transformed into a female sex hormone, flavoring). Estrogen is able to cope with this disease, to prevent or reverse the development of gynecomastia.
In rare cases, the drug Clomiphene Citrate is used as an anabolic agent. The fact that the anti-estrogen has anabolic effect, though not so strong as that of steroids. As already noted, Clomid (Clomiphene) increases the secretion of LH and FSH. These gonadotropins affect the testicles, thereby increasing the level of testosterone in the male and muscle development is observed.
Clomiphene: instructions for use and tips on using
If we talk about the course of preparation, the first and foremost it is worth noting that its use for medical purposes differs from the circuit (dosage, duration of administration, etc.), its use in power sports.
As already noted, clomiphene citrate to treat infertility begins only after a woman will take a full medical examination. Clomiphene is powerful enough, however, in most cases already ovulation occurs on day 5-10 after use of the drug. In medical applications this antiestrogen often take a dose of 50 mg per day.
Application of Clomiphene Citrate is carried out for an average of five days. Before the use of the drug is mandatory stipulate all the details with your doctor. Since the dose and use of the drug in general scheme may differ from the above description.
The use of clomiphene citrate in bodybuilding – a process no less complicated, if not dependent on the individual characteristics of an athlete. Eat Clomid, regardless of your weight and other factors, it should be once a day. Increased frequency of dosing is inappropriate.
The optimum dosage of clomiphene citrate for athletes is on the border of 50-100 micrograms. Even the lowest dose of 50 mg ensure blocking the activity of female hormones and have a positive impact on increasing the level of testosterone. Therefore, to use the drug to the maximum permitted amount of 100 micrograms, is not mandatory.
Clomiphene Citrate Instructions You do not say, but remember that the course of medication should not last longer than 3 weeks. On average, athletes use this anti-estrogen for 2-3 weeks total. This period is sufficient for the manifestation of the effects of the drug (to prevent gynecomastia and rollback and to increase the level of testosterone).